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SGC-CBP30
| Product Name | SGC-CBP30 |
| Price: | Inquiry |
| Catalog No.: | CN00160 |
| CAS No.: | 1613695-14-9 |
| Molecular Formula: | C28H33ClN4O3 |
| Molecular Weight: | 509.04 g/mol |
| Purity: | >=98% |
| Type of Compound: | Alkaloids |
| Physical Desc.: | Powder |
| Source: | |
| Solvent: | Chloroform, Dichloromethane, Ethyl Acetate, DMSO, Acetone, etc. |
| SMILES: | COc1ccc(cc1Cl)CCc1nc2c(n1C[C@@H](N1CCOCC1)C)ccc(c2)c1c(C)noc1C |
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| Description | SGC-CBP30 is a potent CREBBP/EP300 bromodomain inhibitor with IC50 of 21-69 and 38 nM for CREBBP and EP300 bromodomains, respectively.IC50 Value: 21-69 nM(for CREBBP); 38 nM(for EP300)Target: Othersin vivo: SGC-CBP30 is a highly potent and selective p300/CBP bromodomain inhibitor (IC50 ~0.021-0.069 uM for CBP and ~0.038 uM for p300). It has 40-fold selectivity for CBP over BRD4. It accelerated FRAP recovery at 1 uM. in vivo: N/A |
| Density | 1.3±0.1 g/cm3 |
| Boiling Point | 678.0±55.0 °C at 760 mmHg |
| Flash Point | 363.8±31.5 °C |
| Exact Mass | 508.224121 |
| PSA | 65.55000 |
| LogP | 5.29 |
| Vapour Pressure | 0.0±2.1 mmHg at 25°C |
| Storage condition | 2-8°C |